SCHEMBL16612943

SCHEMBL16612943

COc1cccc(CCn2c[c]c(C(N)=O)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.47
NR3C2 P08235 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 1/20 0.42
DAO P14920 1/20 0.42
PARP1 P09874 1/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
AOC3 Q16853 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612857 0.84 MTNR1A (0.44) HRH3MTNR1AMTNR1BPARP1
SCHEMBL16612728 0.82 NR3C2 (0.43) NR3C2TAAR1DAOPARP1MAOB
SCHEMBL16612770 0.76 ADRB2 (0.44) MTNR1AMTNR1B
SCHEMBL12479180 0.76 MTNR1A (0.55) HRH3MTNR1AMTNR1B
SCHEMBL15520091 0.75 CACNA1G (0.43) HDAC1PARP1
SCHEMBL16612868 0.74 MTNR1A (0.49) MTNR1AMTNR1BHDAC1MAOAMAOB
SCHEMBL16612866 0.73 HCRTR2 (0.41) NR3C2
SCHEMBL16612856 0.73 MTNR1A (0.54) MTNR1AMTNR1B
SCHEMBL16612828 0.72 SIRT2 (0.39) HDAC1PARP1MAOBHDAC6
SCHEMBL16612936 0.72 MTNR1A (0.50) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed