SCHEMBL16612828

SCHEMBL16612828

NC(=O)c1[c]cn(CCOc2cccc(F)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.39
HCRTR2 O43614 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
USP2 O75604 1/20 0.38
KMT2A Q03164 1/20 0.38
MAOB P27338 1/20 0.38
PARP10 Q53GL7 1/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
GRM5 P41594 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36
ICMT O60725 1/20 0.36
HPGDS O60760 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612857 0.86 MTNR1A (0.44) KMT2ALMNASMN1; SMN2HTR1ADRD2
SCHEMBL16612775 0.85 MAOB (0.41) MAOBPARP10SMN1; SMN2
SCHEMBL16612728 0.80 NR3C2 (0.43) MAOBPARP10PARP1
SCHEMBL15520701 0.77 L3MBTL1 (0.50) KMT2AMAOBPARP10SMN1; SMN2NPSR1
SCHEMBL16612880 0.76 DRD2 (0.45) HCRTR2KMT2AMAOBLMNASMN1; SMN2
SCHEMBL16612782 0.74 HCRTR2 (0.39) HCRTR2HTR1AHTR7GRM5PARP1
SCHEMBL16612665 0.74 HCRTR2 (0.39) HCRTR2
SCHEMBL16613032 0.73 HCRTR2 (0.44) HCRTR2
SCHEMBL16612990 0.72 HCRTR2 (0.39) HCRTR2
SCHEMBL16612943 0.72 SIGMAR1 (0.47) MAOBHDAC6HDAC1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed