SCHEMBL16612786

SCHEMBL16612786

Cn1nc(OCCn2c[c]c(C(N)=O)n2)cc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
NPC1 O15118 1/20 0.41
HCRTR2 O43614 1/20 0.41
RAB9A P51151 1/20 0.40
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612935 0.76 HCRTR2 (0.38) HCRTR2KMT2A
SCHEMBL16612990 0.76 HCRTR2 (0.39) PKMHCRTR2ALDH1A1
SCHEMBL16613011 0.74 HCRTR2 (0.36) HCRTR2
SCHEMBL16612850 0.74 HCRTR2 (0.38) HCRTR2MAPTSMN1; SMN2ALDH1A1
SCHEMBL16612712 0.74 HCRTR2 (0.38) HCRTR2SMN1; SMN2ALDH1A1GAA
SCHEMBL16612782 0.74 HCRTR2 (0.39) HCRTR2
SCHEMBL16612877 0.72 HCRTR2 (0.35) HCRTR2
SCHEMBL16612787 0.71 PKM (0.49) PKMNPC1HCRTR2RAB9AMAPT
SCHEMBL16612857 0.71 MTNR1A (0.44) PKMNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL16612828 0.71 SIRT2 (0.39) HCRTR2SMN1; SMN2NPSR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed