SCHEMBL16612990

SCHEMBL16612990

Cc1ccnc(OCCn2c[c]c(C(N)=O)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 4/20 0.39
HCRTR1 O43613 3/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
JMJD6 Q6NYC1 3/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
PKM P14618 1/20 0.31
PLAU P00749 1/20 0.31
PPARG P37231 1/20 0.31
CCR1 P32246 1/20 0.30
CCR5 P51681 1/20 0.30
CCR8 P51685 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612935 0.84 HCRTR2 (0.38) HCRTR2HCRTR1
SCHEMBL16612850 0.82 HCRTR2 (0.38) HCRTR2HCRTR1ALDH1A1
SCHEMBL16612782 0.79 HCRTR2 (0.39) HCRTR2HCRTR1PPARG
SCHEMBL16612877 0.78 HCRTR2 (0.35) HCRTR2
SCHEMBL16612786 0.76 PKM (0.54) HCRTR2PKMALDH1A1
SCHEMBL16612712 0.75 HCRTR2 (0.38) HCRTR2HCRTR1ALDH1A1
SCHEMBL16613011 0.75 HCRTR2 (0.36) HCRTR2HCRTR1
SCHEMBL16612857 0.74 MTNR1A (0.44) PKMALDH1A1
SCHEMBL16613039 0.74 MEN1 (0.46) HCRTR2HCRTR1ALDH1A1
SCHEMBL16612828 0.72 SIRT2 (0.39) HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed