SCHEMBL16612935

SCHEMBL16612935

Cc1cc(C)nc(OCCn2c[c]c(C(N)=O)n2)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.38
HCRTR1 O43613 1/20 0.38
POLQ O75417 1/20 0.35
IKBKB O14920 3/20 0.31
SYK P43405 2/20 0.31
KCNH2 Q12809 2/20 0.31
GRM5 P41594 1/20 0.31
THRB P10828 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612782 0.84 HCRTR2 (0.39) HCRTR2HCRTR1GRM5
SCHEMBL16612990 0.84 HCRTR2 (0.39) HCRTR2HCRTR1
SCHEMBL16612850 0.80 HCRTR2 (0.38) HCRTR2HCRTR1
SCHEMBL16612877 0.78 HCRTR2 (0.35) HCRTR2SYK
SCHEMBL16612712 0.78 HCRTR2 (0.38) HCRTR2HCRTR1
SCHEMBL16612786 0.76 PKM (0.54) HCRTR2KMT2A
SCHEMBL16613039 0.74 MEN1 (0.46) HCRTR2HCRTR1KMT2A
SCHEMBL16613011 0.73 HCRTR2 (0.36) HCRTR2HCRTR1GRM5
SCHEMBL16612772 0.72 KMT2A (0.46) HCRTR2HCRTR1SYKKMT2A
SCHEMBL16612857 0.72 MTNR1A (0.44) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed