SCHEMBL16612856

SCHEMBL16612856

COc1ccc2ncn(CCn3c[c]c(C(N)=O)n3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.54
MTNR1B P49286 3/20 0.54
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
CDYL2 Q8N8U2 1/20 0.39
CDYL Q9Y232 1/20 0.39
CDY1; CDY1B Q9Y6F8 1/20 0.39
MAPT P10636 1/20 0.39
TBXA2R P21731 1/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPK10 P53779 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
P2RX3 P56373 2/20 0.38
KDM4E B2RXH2 2/20 0.37
PLK1 P53350 4/20 0.37
NEK2 P51955 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16613026 0.85 HDAC6 (0.40) MTNR1AMTNR1BHCRTR2PLK1
SCHEMBL16612854 0.82 MTNR1A (0.52) MTNR1AMTNR1BHCRTR1HCRTR2HTT
SCHEMBL16612739 0.81 TDP1 (0.54) HTTALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL16612868 0.81 MTNR1A (0.49) MTNR1AMTNR1BHCRTR1HCRTR2ALDH1A1
SCHEMBL16612936 0.76 MTNR1A (0.50) MTNR1AMTNR1BHCRTR2
SCHEMBL16612997 0.76 HCRTR2 (0.42) MTNR1AMTNR1BHCRTR1HCRTR2HTT
SCHEMBL27038883 0.76 MTNR1A (0.65) MTNR1AMTNR1BHCRTR1HCRTR2CDYL2
SCHEMBL16612857 0.75 MTNR1A (0.44) MTNR1AMTNR1BALDH1A1MAPK1MAPK10
SCHEMBL16612770 0.74 ADRB2 (0.44) MTNR1AMTNR1BHCRTR1HCRTR2ALDH1A1
SCHEMBL12479232 0.73 MTNR1A (0.66) MTNR1AMTNR1BCDYL2CDYLCDY1; CDY1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed