SCHEMBL16612936

SCHEMBL16612936

COc1ccc2ccn(CCCn3c[c]c(C(N)=O)n3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.50
MTNR1B P49286 6/20 0.50
MCL1 Q07820 8/20 0.48
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
TRPV1 Q8NER1 1/20 0.43
HCRTR2 O43614 1/20 0.42
HTR7 P34969 1/20 0.41
ADA P00813 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612854 0.94 MTNR1A (0.52) MTNR1AMTNR1BMCL1HTR2AHTR2C
SCHEMBL16612868 0.86 MTNR1A (0.49) MTNR1AMTNR1BHTR2AHTR2CHCRTR2
SCHEMBL16612920 0.84 CDK4 (0.52) MTNR1AMTNR1B
SCHEMBL16612831 0.80 HCRTR2 (0.42) MTNR1AMTNR1BHCRTR2
SCHEMBL16612997 0.78 HCRTR2 (0.42) MTNR1AMTNR1BMCL1HCRTR2
SCHEMBL16612628 0.78 HCRTR2 (0.43) MTNR1AMTNR1BMCL1HCRTR2
SCHEMBL16612876 0.78 HTR2C (0.41) MTNR1AMTNR1BHTR2AHTR2CHCRTR2
SCHEMBL16612954 0.77 LMNA (0.53) MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL16612656 0.77 HCRTR2 (0.42) MTNR1AMTNR1BHCRTR2
SCHEMBL16612856 0.76 MTNR1A (0.54) MTNR1AMTNR1BHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed