SCHEMBL16612997

SCHEMBL16612997

COc1cc(OC)c2ccn(CCn3c[c]c(C(N)=O)n3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.42
HCRTR1 O43613 1/20 0.42
HTR6 P50406 1/20 0.38
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
MTNR1A P48039 6/20 0.34
MTNR1B P49286 6/20 0.34
ABCG2 Q9UNQ0 2/20 0.33
PDE10A Q9Y233 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
TRPM5 Q9NZQ8 2/20 0.33
MCL1 Q07820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612854 0.83 MTNR1A (0.52) HCRTR2HCRTR1NPC1RAB9AALDH1A1
SCHEMBL16612868 0.82 MTNR1A (0.49) HCRTR2HCRTR1NPC1RAB9AALDH1A1
SCHEMBL16612831 0.82 HCRTR2 (0.42) HCRTR2HCRTR1MTNR1AMTNR1BTSHR
SCHEMBL16613148 0.81 HCRTR2 (0.42) HCRTR2MTNR1AMTNR1B
SCHEMBL16612656 0.79 HCRTR2 (0.42) HCRTR2HCRTR1MTNR1AMTNR1BTSHR
SCHEMBL16612960 0.78 HCRTR2 (0.41) HCRTR2TRPM5
SCHEMBL16612936 0.78 MTNR1A (0.50) HCRTR2MTNR1AMTNR1BMCL1
SCHEMBL16612856 0.76 MTNR1A (0.54) HCRTR2HCRTR1ALDH1A1HPGDMTNR1A
SCHEMBL16612628 0.76 HCRTR2 (0.43) HCRTR2HCRTR1MTNR1AMTNR1BMCL1
SCHEMBL16613000 0.75 HTR2A (0.42) HCRTR2HCRTR1LMNAMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed