SCHEMBL16623552

SCHEMBL16623552

Cc1c[nH]c(=O)c(C(=N)C2CC2)c1Nc1c(F)cccc1F

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
HDAC4 P56524 1/20 0.32
BRD4 O60885 2/20 0.32
CREBBP Q92793 2/20 0.32
GAA P10253 2/20 0.31
MAPT P10636 1/20 0.31
ABL1 P00519 2/20 0.31
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
JAK3 P52333 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849204 0.86 GAA (0.36) DDB1CRBNHDAC4GAAJAK2
SCHEMBL17849219 0.73 RAF1 (0.42) GAAMAPT
SCHEMBL16623479 0.73 CRBN (0.40) CRBNBRD4CREBBP
SCHEMBL16623480 0.73 MAPK14 (0.34)
SCHEMBL16623554 0.73 MAPK14 (0.33) JAK2JAK1JAK3
SCHEMBL16623594 0.69 CMA1 (0.35)
SCHEMBL17849236 0.62 RORC (0.36) GAA
SCHEMBL16726675 0.61
SCHEMBL17849237 0.61 RORC (0.33)
SCHEMBL24237192 0.61 ACHE (0.50) HDAC4MAPTJAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed