SCHEMBL1662873

SCHEMBL1662873

COc1ccc(N2CCN(C(=O)OC(C)(C)C)CC2=O)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.47
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
ALDH1A1 P00352 1/20 0.45
RBP4 P02753 1/20 0.44
ESR2 Q92731 1/20 0.42
STS P08842 1/20 0.41
NR1H2 P55055 1/20 0.41
NPY2R P49146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1584703 0.87 CPS1 (0.46) P2RX7KDM4EMAPTALDH1A1STS
SCHEMBL1663013 0.82 P2RX7 (0.56) P2RX7RBP4
SCHEMBL1665532 0.81 ALDH1A1 (0.53) KDM4EMAPTALDH1A1STSNR1H2
SCHEMBL31342592 0.78 SUV39H2 (0.44) P2RX7MAPTALDH1A1RBP4ESR2
SCHEMBL2366725 0.77 NR1H2 (0.44) P2RX7MAPTALDH1A1ESR2NR1H2
SCHEMBL1662799 0.76 NR1H2 (0.41) P2RX7KDM4EMAPTALDH1A1RBP4
SCHEMBL1583767 0.76 GPR119 (0.46) KDM4EMAPTALDH1A1NR1H2
SCHEMBL4537183 0.76 P2RX7 (0.55) P2RX7
SCHEMBL22650493 0.75 NR1H2 (0.54) P2RX7ESR2NR1H2
SCHEMBL1662960 0.75 P2RX7 (0.44) P2RX7MAPTESR2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050284-A1 PYRAZOLYLPYRIDINE ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2011-04-28 WO disclosed