SCHEMBL16634644

SCHEMBL16634644

NC(=NO)c1ccc(-n2c(=O)n(C(=O)c3c(Cl)cccc3Cl)c3ccccc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 9/20 0.40
CYP2C9 P11712 5/20 0.35
CYP3A4 P08684 4/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 2/20 0.35
RARG P13631 1/20 0.35
FFAR2 O15552 1/20 0.34
HPGD P15428 3/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GAA P10253 2/20 0.32
GFER P55789 1/20 0.32
NPC1 O15118 2/20 0.32
GLA P06280 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TSHR P16473 1/20 0.32
PKM P14618 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634830 0.88 RORC (0.43) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634554 0.84 RORC (0.55) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634709 0.80 TAS1R3 (0.44) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634643 0.80 RORC (0.40) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634740 0.78 RORC (0.37) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634721 0.77 RAB9A (0.45) RORCRAB9ASMN1; SMN2NPC1TSHR
SCHEMBL16634636 0.75 RORC (0.56) RORCCYP2C9CYP3A4CYP2C19
SCHEMBL16634666 0.74 MYC (0.48) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634717 0.72 RORC (0.55) RORCCYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL16634779 0.72 RORC (0.53) RORCCYP2C9CYP3A4CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed