SCHEMBL16634724

SCHEMBL16634724

O=C(O)c1ccc(-n2c(=O)[nH]c3cnccc32)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
PARP1 P09874 1/20 0.45
CSNK2A1 P68400 1/20 0.45
AURKA O14965 2/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
DAO P14920 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
TNKS O95271 1/20 0.37
CSNK2A2 P19784 2/20 0.37
CSNK2B P67870 2/20 0.37
B3GNT2 Q9NY97 2/20 0.37
FEN1 P39748 1/20 0.36
RORC P51449 1/20 0.36
HSP90AA1 P07900 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634626 0.83 HSP90AA1 (0.54) CYP3A4PARP1AURKAKDM4ESMN1; SMN2
SCHEMBL15552842 0.81 TGFBR1 (0.52) TGFBR1CYP1A2CYP3A4PARP1DAO
SCHEMBL16657405 0.80 TNKS (0.51) PARP1CSNK2A1AURKAKDM4EDAO
SCHEMBL16657401 0.79 TGFBR1 (0.47) TGFBR1CYP1A2CYP3A4KDM4ETNKS
SCHEMBL16634859 0.77 AURKA (0.44) CYP1A2CYP3A4CSNK2A1AURKAKDM4E
SCHEMBL16634608 0.76 RORC (0.47) AURKAKDM4ESMN1; SMN2DAOSLC22A12
SCHEMBL16634734 0.74 DAO (0.50) CYP3A4AURKAKDM4ESMN1; SMN2DAO
SCHEMBL30615562 0.74 TGFBR1 (0.48) TGFBR1CYP1A2CYP3A4KDM4ETNKS
SCHEMBL21463483 0.74 TGFBR1 (0.48) TGFBR1CYP1A2CYP3A4KDM4ETNKS
SCHEMBL30615513 0.72 TGFBR1 (0.54) TGFBR1CYP1A2CYP3A4DAOTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed