SCHEMBL16634626

SCHEMBL16634626

O=C(O)c1ccc(-n2c(=O)[nH]c3ccccc32)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.54
AURKA O14965 2/20 0.52
KDM4E B2RXH2 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
RORC P51449 3/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
HSD11B1 P28845 1/20 0.43
B3GNT2 Q9NY97 2/20 0.42
DAO P14920 1/20 0.42
GABRP O00591 2/20 0.42
GABRD O14764 2/20 0.42
GABRA1 P14867 2/20 0.42
GABRB1 P18505 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA5 P31644 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634734 0.83 DAO (0.50) AURKAKDM4ESMN1; SMN2RORCCYP3A4
SCHEMBL16634724 0.83 TGFBR1 (0.47) HSP90AA1AURKAKDM4ESMN1; SMN2RORC
SCHEMBL21463543 0.82 HSP90AA1 (0.57) HSP90AA1AURKADAOGABRPGABRD
SCHEMBL30615631 0.82 HSP90AA1 (0.57) HSP90AA1AURKADAOGABRPGABRD
SCHEMBL16634859 0.81 AURKA (0.44) HSP90AA1AURKAKDM4ESMN1; SMN2CYP3A4
SCHEMBL16634608 0.80 RORC (0.47) AURKAKDM4ESMN1; SMN2RORCCYP2C9
SCHEMBL23119726 0.80 HSP90AA1 (0.56) HSP90AA1AURKAKDM4EDAOGABRP
SCHEMBL22583745 0.80 AURKA (0.55) HSP90AA1AURKADAOGABRPGABRD
SCHEMBL5011347 0.78 KDM4E (0.78) AURKAKDM4ESMN1; SMN2PARP1
SCHEMBL16634744 0.77 L3MBTL1 (0.55) HSP90AA1AURKAKDM4ESMN1; SMN2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed