SCHEMBL16634734

SCHEMBL16634734

O=C(O)c1ccc(-n2c(=O)[nH]c3cccc(F)c32)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.50
KDM4E B2RXH2 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RORC P51449 8/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 1/20 0.44
AURKA O14965 2/20 0.43
TTR P02766 1/20 0.40
FEN1 P39748 1/20 0.39
B3GNT2 Q9NY97 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634626 0.83 HSP90AA1 (0.54) DAOKDM4ESMN1; SMN2RORCCYP3A4
SCHEMBL16634793 0.83 DAO (0.43) DAOKDM4ESMN1; SMN2CYP3A4CYP2C9
SCHEMBL16634608 0.79 RORC (0.47) DAOKDM4ESMN1; SMN2RORCCYP2C9
SCHEMBL5011347 0.74 KDM4E (0.78) KDM4ESMN1; SMN2AURKA
SCHEMBL16634724 0.74 TGFBR1 (0.47) DAOKDM4ESMN1; SMN2RORCCYP3A4
SCHEMBL16634795 0.74 DAO (0.44) DAOFEN1
SCHEMBL16634859 0.72 AURKA (0.44) KDM4ESMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL16634752 0.68 RORC (0.56) RORCCYP3A4CYP2C9CYP2C19
SCHEMBL5011339 0.65 KDM4E (0.59) KDM4ESMN1; SMN2
SCHEMBL21491217 0.65 BCAT1 (0.55) KDM4ESMN1; SMN2CYP2C9CYP2C19TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed