SCHEMBL1665086

SCHEMBL1665086

CCC(C)(C)C(=O)SCCC(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.44
HSD17B10 Q99714 3/20 0.37
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 3/20 0.34
CA12 O43570 2/20 0.34
CA14 Q9ULX7 2/20 0.34
KDM4E B2RXH2 1/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 3/20 0.33
PTGS1 P23219 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
TET2 Q6N021 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10085341 0.91 TSHR (0.47) TSHRHSD17B10KMT2AMEN1LMNA
SCHEMBL10085230 0.83 CYP1A2 (0.41) TSHRKMT2AMEN1LMNAKDM4E
SCHEMBL1665311 0.82 TSHR (0.36) TSHRHSD17B10KMT2AMEN1KDM4E
SCHEMBL6891006 0.80 TSHR (0.42) TSHRHSD17B10KMT2AMEN1LMNA
SCHEMBL14566406 0.78 MEN1 (0.33) KMT2AMEN1ALDH1A1
SCHEMBL12149865 0.75 RIPK1 (0.31) KDM4E
SCHEMBL17403974 0.74 ACHE (0.38)
SCHEMBL13522419 0.74 RIPK1 (0.31)
SCHEMBL12695618 0.74 NOS3 (0.40) HSD17B10ALDH1A1MAPT
SCHEMBL9509274 0.73 TSHR (0.55) TSHRHSD17B10KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 125 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12371723-B2 Variant LovD polypeptides and their uses CODEXIS, INC. (US) 2025-07-29 US disclosed
US-20240368649-A1 LOV-D ACYLTRANSFERASE MEDIATED ACYLATION CODEXIS INC (US) 2024-11-07 US disclosed
US-12060592-B2 Lov-D acyltransferase mediated acylation CODEXIS, INC. (US) 2024-08-13 US disclosed
US-20240218407-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2024-07-04 US disclosed
US-20240218407-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2024-07-04 US disclosed
US-20240218407-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2024-07-04 US disclosed
US-11926857-B2 Variant LovD polypeptides and their uses CODEXIS, INC. (US) 2024-03-12 US disclosed
US-20210277432-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2021-09-09 US disclosed
US-20210277432-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2021-09-09 US disclosed
US-11046982-B2 Variant LovD polypeptides and their uses CODEXIS, INC. (US) 2021-06-29 US disclosed
EP-2032715-B1 Methods and materials for making simvastatin and related compounds UNIV CALIFORNIA (US) 2012-02-01 EP disclosed
US-20110111468-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES CODEXIS, INC. (US) 2011-05-12 US disclosed
US-20110111468-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES CODEXIS, INC. (US) 2011-05-12 US disclosed
US-20110111468-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES CODEXIS, INC. (US) 2011-05-12 US disclosed
WO-2011041231-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES CODEXIS, INC. (US) 2011-04-07 WO disclosed
WO-2011041231-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES CODEXIS, INC. (US) 2011-04-07 WO disclosed
WO-2011041233-A1 IMPROVED LOV-D ACYLTRANSFERASE MEDIATED ACYLATION CODEXIS, INC. (US) 2011-04-07 WO disclosed
WO-2011041233-A1 IMPROVED LOV-D ACYLTRANSFERASE MEDIATED ACYLATION CODEXIS, INC. (US) 2011-04-07 WO disclosed
US-20090191602-A1 Methods and Materials for Making Simvastatin and Related Compounds INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2009-07-30 US disclosed
US-20090191602-A1 Methods and Materials for Making Simvastatin and Related Compounds INNOVATUS LIFE SCIENCES LENDING FUND I, LP, AS COLLATERAL AGENT 2009-07-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240368649-A1 LOV-D ACYLTRANSFERASE MEDIATED ACYLATION ACAT2, LCAT, ACOT7 TSHR 4462/4885HSD17B10 118/4885KMT2A 579/4885
US-11046982-B2 Variant LovD polypeptides and their uses LCAT, HMGCR, FNTA TSHR 4500/4885HSD17B10 66/4885KMT2A 2211/4885
US-12060592-B2 Lov-D acyltransferase mediated acylation ACAT2, LCAT, ACOT7 TSHR 4462/4885HSD17B10 118/4885KMT2A 579/4885
US-20210277432-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES LCAT, HMGCR, FNTA TSHR 4500/4885HSD17B10 66/4885KMT2A 2211/4885
US-11926857-B2 Variant LovD polypeptides and their uses LCAT, HMGCR, FNTA TSHR 4500/4885HSD17B10 66/4885KMT2A 2211/4885
US-20110111468-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES PCSK9, HMGCR, LCAT TSHR 4517/4885HSD17B10 67/4885KMT2A 2868/4885
US-20240218407-A1 VARIANT LOVD POLYPEPTIDES AND THEIR USES LCAT, HMGCR, FNTA TSHR 4500/4885HSD17B10 66/4885KMT2A 2211/4885
US-12371723-B2 Variant LovD polypeptides and their uses LCAT, HMGCR, FNTA TSHR 4500/4885HSD17B10 66/4885KMT2A 2211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.