SCHEMBL16664924

SCHEMBL16664924

CC(C)(C)CNc1cc(-c2ccc(NC3CCN(C4CC4)CC3)nc2)ncn1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.41
HRH3 Q9Y5N1 2/20 0.40
SYK P43405 6/20 0.38
TBK1 Q9UHD2 1/20 0.37
IRAK4 Q9NWZ3 2/20 0.37
TDO2 P48775 1/20 0.37
ACKR3 P25106 1/20 0.37
RORC P51449 1/20 0.37
PIK3CD O00329 1/20 0.36
CCR6 P51684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15343201 0.90 PIK3CA (0.41) HRH3SYKTBK1IRAK4TDO2
SCHEMBL19355418 0.80 CYP1A2 (0.46) SYK
SCHEMBL16664942 0.79 SYK (0.49) HRH4SYKTBK1TDO2
SCHEMBL17634513 0.79 CYP1A2 (0.41) SYKIRAK4
SCHEMBL19905357 0.76 CYP2D6 (0.39) SYKIRAK4
SCHEMBL16664930 0.76 GPR39 (0.42) HRH4HRH3
SCHEMBL16665019 0.76 TDO2 (0.44) SYKTBK1TDO2CCR6
SCHEMBL16660261 0.75 PIK3CA (0.46) HRH4
SCHEMBL19819913 0.75 HPGDS (0.44) HRH4SYKTBK1TDO2
SCHEMBL19905240 0.74 SYK (0.41) HRH4SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed