SCHEMBL1670782

SCHEMBL1670782

COc1ccc(-c2c[nH]c(C#N)c2N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.44
MAPT P10636 6/20 0.43
PTPN1 P18031 2/20 0.43
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPKAPK2 P49137 1/20 0.42
ALDH1A1 P00352 5/20 0.41
HPGD P15428 4/20 0.41
KDM4E B2RXH2 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800387 0.78 MAPT (0.53) MAPTKMT2AALDH1A1HPGDKDM4E
SCHEMBL22283897 0.78 ADORA1 (0.51) ADORA1MAPTPTPN1PRKAB2PRKAG1
SCHEMBL1185412 0.78 ALDH1A1 (0.51) ADORA1MAPTPTPN1PRKAB2PRKAG1
SCHEMBL7689092 0.70 POLB (0.49) ADORA1MAPTPTPN1MEN1KMT2A
SCHEMBL12670739 0.69 PRKAB2 (0.51) ADORA1MAPTPRKAB2PRKAG1PRKAA2
SCHEMBL140629 0.69 PGR (0.49) ADORA1MAPTPTPN1PRKAB2PRKAG1
SCHEMBL11021063 0.69 PIM1 (0.49) MAPTPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL21608938 0.69 ALDH1A1 (0.54) ADORA1MAPTPTPN1MEN1KMT2A
SCHEMBL7574828 0.69 KMT2A (0.55) ADORA1MAPTPTPN1MEN1KMT2A
SCHEMBL1670787 0.68 MAPKAPK2 (0.47) ADORA1MAPTPTPN1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed