SCHEMBL1670823

SCHEMBL1670823

O=C(CCOCCCNC(=O)c1ccc(O)c(C2(c3ccccc3)CCNCC2)c1)OC(=O)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
PDK2 Q15119 2/20 0.35
TACR1 P25103 1/20 0.35
ITGA2 P17301 1/20 0.34
HPGD P15428 2/20 0.34
MAPT P10636 3/20 0.34
NAMPT P43490 2/20 0.33
MLYCD O95822 2/20 0.33
PRSS1 P07477 1/20 0.33
CTSG P08311 1/20 0.33
CTRB1 P17538 1/20 0.33
CMA1 P23946 1/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670831 0.96 SMN1; SMN2 (0.36) ITGB3ITGA2BPDK2TACR1ITGA2
Trifluoroacetic Acid SCHEMBL1670822 0.89 ITGB3 (0.42) ITGB3ITGA2BPDK2TACR1ITGA2
Trifluoroacetic Acid SCHEMBL1670826 0.85 ITGB3 (0.41) ITGB3ITGA2BPDK2TACR1ITGA2
SCHEMBL1668840 0.76 NAMPT (0.42) HPGDMAPTNAMPTTP53
SCHEMBL12801195 0.76 KDM4E (0.42) TACR1NAMPTHDAC1
SCHEMBL1668619 0.72 FFAR4 (0.35) TACR1
SCHEMBL12800770 0.70 OPRD1 (0.42) TACR1MAPTNAMPTHDAC1HTT
SCHEMBL1670835 0.70 OPRM1 (0.43) MAPTNAMPTTP53HDAC1HTT
SCHEMBL1669606 0.69 CA12 (0.47) PDK2HPGDMAPTTP53HDAC1
SCHEMBL12800418 0.68 OPRM1 (0.40) ITGB3ITGA2BTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed