SCHEMBL1671018

SCHEMBL1671018

Cc1noc(C)c1-c1c(Br)cn(C)c1C#N

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.36
BRD2 P25440 2/20 0.36
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
TLR8 Q9NR97 1/20 0.33
USP30 Q70CQ3 4/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
AR P10275 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
USP2 O75604 1/20 0.31
BRD3 Q15059 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800965 0.77 TLR8 (0.40) BRD4BRD2CYP3A4CYP2D6CYP2C19
SCHEMBL1670383 0.75 BRD4 (0.40) BRD4BRD2USP30AR
SCHEMBL1670709 0.73 PTGS2 (0.48) BRD4BRD2NPSR1BRD3
SCHEMBL1670817 0.69 MLYCD (0.40) BRD4BRD2USP30AR
SCHEMBL16411423 0.68 HDAC8 (0.32)
SCHEMBL1673047 0.66 IMPDH2 (0.31)
SCHEMBL1682484 0.64 BRD4 (0.40) BRD4BRD2USP30AR
SCHEMBL25975652 0.62 BRD4 (0.59) BRD4BRD2USP30ARBRD3
SCHEMBL15106914 0.60 TLR8 (0.45) BRD4BRD2CYP3A4CYP2C19TLR8
SCHEMBL18812499 0.59 BRD4 (0.51) BRD4BRD2CYP3A4ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed