SCHEMBL1670709

SCHEMBL1670709

COc1ccc(-c2cn(C)c(C#N)c2-c2c(C)noc2C)cc1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.48
BRD4 O60885 12/20 0.46
CREBBP Q92793 1/20 0.41
BRD2 P25440 3/20 0.40
BRD3 Q15059 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670383 0.86 BRD4 (0.40) BRD4CREBBPBRD2
SCHEMBL12800381 0.82 PTGS2 (0.51) PTGS2BRD4BRD2BRD3
SCHEMBL1670920 0.81 PTGS2 (0.47) PTGS2BRD4CREBBPBRD2BRD3
SCHEMBL17833811 0.76 PTGS2 (0.72) PTGS2BRD4BRD2BRD3
SCHEMBL1671018 0.73 BRD4 (0.36) BRD4BRD2BRD3NPSR1
SCHEMBL1670381 0.72 MAPKAPK2 (0.41) NPSR1
SCHEMBL1670787 0.72 MAPKAPK2 (0.47) NPSR1
SCHEMBL12800374 0.69 PTGS2 (0.50) PTGS2BRD4BRD2BRD3
SCHEMBL1670583 0.68 MAOA (0.38) PTGS2BRD4
SCHEMBL1653145 0.68 BRD4 (0.48) PTGS2BRD4CREBBPBRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed