Cyclohexyl(Hydroxy)Methylenediphosphonic Acid

Cyclohexyl(Hydroxy)Methylenediphosphonic Acid

SCHEMBL1674148

O=P(O)(O)C(O)(C1CCCCC1)P(=O)(O)O

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FDPS P14324 3/20 0.37
MMP2 P08253 7/20 0.35
CA12 O43570 6/20 0.35
CA1 P00915 6/20 0.35
CA2 P00918 6/20 0.35
CA9 Q16790 6/20 0.35
MMP1 P03956 3/20 0.35
MMP8 P22894 2/20 0.35
MMP3 P08254 2/20 0.35
METAP1 P53582 1/20 0.35
MMP9 P14780 1/20 0.32
LMNA P02545 1/20 0.32
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
ANPEP P15144 2/20 0.31
ERAP2 Q6P179 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055491 0.82 CA12 (0.32) FDPSMMP2CA12CA1CA2
SCHEMBL12076033 0.80 FDPS (0.37) FDPSMMP2CA12CA1CA2
SCHEMBL6352733 0.77 MMP2 (0.37) FDPSMMP2CA12CA1CA2
SCHEMBL10341430 0.76 ALDH1A1 (0.32) FDPS
SCHEMBL9806690 0.76 LMNA (0.38) FDPSLMNAANPEPERAP2
SCHEMBL8055401 0.76 MMP2 (0.33) FDPSMMP2CA12CA1CA2
SCHEMBL10384523 0.74 SLC6A1 (0.38) FDPSLMNA
SCHEMBL3794209 0.73 METAP1 (0.38) FDPSMMP2CA12CA1CA2
SCHEMBL27864692 0.73 LMNA (0.36) FDPSMMP2CA12CA1CA2
SCHEMBL4088811 0.73 METAP1 (0.38) FDPSMMP2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3194505-B1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INT AG (CH) 2022-03-02 EP claimed
US-20170275175-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INTERNATIONAL AG (CH) 2017-09-28 US claimed
EP-3194505-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL Omya International AG (CH) 2017-07-26 EP claimed
WO-2016041781-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INTERNATIONAL AG (CH) 2016-03-24 WO claimed
EP-2995654-A1 Dry process for preparing a surface-modified alkaline earth metal carbonate-containing material Omya International AG (CH) 2016-03-16 EP claimed
EP-0563096-B1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 2000-05-03 EP claimed
EP-0563096-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1993-10-06 EP claimed
EP-3194505-B1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INT AG (CH) 2022-03-02 EP disclosed
US-10836646-B2 Dry process for preparing a surface-modified alkaline earth metal carbonate-containing material OMYA INTERNATIONAL AG (US) 2020-11-17 US disclosed
US-20170275175-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INTERNATIONAL AG (CH) 2017-09-28 US disclosed
EP-3194505-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL Omya International AG (CH) 2017-07-26 EP disclosed
WO-2016041781-A1 DRY PROCESS FOR PREPARING A SURFACE-MODIFIED ALKALINE EARTH METAL CARBONATE-CONTAINING MATERIAL OMYA INTERNATIONAL AG (CH) 2016-03-24 WO disclosed
EP-2995654-A1 Dry process for preparing a surface-modified alkaline earth metal carbonate-containing material Omya International AG (CH) 2016-03-16 EP disclosed
WO-1995023510-A1 A METHOD OF INHIBITING THE FORMATION OF CRYSTALLINE MINERAL DEPOSITS IN SOIL CH2O INCORPORATED (US) 1995-09-08 WO disclosed
US-5256653-A Pharmaceutical preparations containing platinum complexes/phosphonic acid liquid and processes for their use HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1993-10-26 US disclosed
EP-0563096-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1993-10-06 EP disclosed
WO-1992011267-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1992-07-09 WO disclosed
EP-0345294-A1 DRUGS CONTAINING PLATINUM COMPLEXES. HENKEL KGAA (DE) 1989-12-13 EP disclosed
US-4802990-A DESCALING WATER SYSTEMS WITH 1, HYDROXYETHANE 1,1-DIPHOSPHONIC ACID; HYDROXYMETHYLENE PHOSPHONIC ACID, POTASSIUM HYDROXIDE; AMMONIA EUGENE L. INSKEEP 1989-02-07 US disclosed
WO-1988006149-A1 PLATINUM COMPLEXES, PROCESS FOR THEIR PRODUCTION AND DRUGS CONTAINING SAME HENKEL KGAA (DE) 1988-08-25 WO disclosed