SCHEMBL16748696

SCHEMBL16748696

CCCCOc1c[nH]c(CNSc2ccc(C(=O)O)cc2)cc1=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PLA2G4B P0C869 4/20 0.43
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
WDR5 P61964 1/20 0.39
PTPN11 Q06124 1/20 0.39
RARB P10826 5/20 0.39
GRM2 Q14416 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
RXRA P19793 1/20 0.37
PLA2G4A P47712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9915516 0.80 PLA2G4B (0.41) PLA2G4BTP53TSHRWDR5PTPN11
SCHEMBL9915532 0.77 HPGD (0.36) ALDH1A1HPGD
SCHEMBL16748804 0.76 NR1H4 (0.46) TP53TSHR
SCHEMBL16748648 0.76 CDK1 (0.38)
SCHEMBL15279055 0.72 CDK1 (0.35) TP53TSHR
SCHEMBL14818596 0.71 CDK1 (0.40) ALDH1A1
SCHEMBL9915471 0.71 SMN1; SMN2 (0.40) TSHRHPGD
SCHEMBL16748830 0.71 CDK1 (0.37) PTPN11
SCHEMBL9915324 0.69 CDK1 (0.38) TP53ALDH1A1
SCHEMBL14136577 0.69 USP2 (0.45) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed