SCHEMBL16748830

SCHEMBL16748830

CCCCOc1c[nH]c(CC(=O)C(=O)O)cc1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.37
CCNB1 P14635 3/20 0.37
CDK2 P24941 3/20 0.37
CDK4 P11802 2/20 0.37
CCND1 P24385 2/20 0.37
CCNT1 O60563 1/20 0.37
CCNA2 P20248 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK9 P50750 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
RB1 P06400 1/20 0.36
CA9 Q16790 1/20 0.35
S1PR3 Q99500 1/20 0.34
XDH P47989 2/20 0.33
PTPN11 Q06124 1/20 0.33
PDE4B Q07343 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14818596 0.81 CDK1 (0.40) CDK1CCNB1CDK2CDK4CCND1
SCHEMBL9915324 0.79 CDK1 (0.38) CDK1CCNB1CDK2CDK4CCND1
SCHEMBL16748648 0.78 CDK1 (0.38) CDK1CCNB1CDK2CDK4CCND1
SCHEMBL15279041 0.76 ALDH1A1 (0.39) GAA
SCHEMBL15279055 0.74 CDK1 (0.35) CDK1CCNB1CDK2CDK4CCND1
SCHEMBL9915516 0.72 PLA2G4B (0.41) PTPN11
SCHEMBL16748696 0.71 PLA2G4B (0.43) PTPN11
SCHEMBL15279003 0.70 DAO (0.43)
SCHEMBL9291158 0.69 GHSR (0.43) S1PR3PDE4BKDM4EMEN1KMT2A
SCHEMBL9915491 0.67 SMYD3 (0.45) PTPN11KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed