SCHEMBL1684142

SCHEMBL1684142

O=C(c1cc2[nH]cnc2cn1)N(O)Cc1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.43
QPCT Q16769 5/20 0.40
QPCTL Q9NXS2 1/20 0.40
HDAC3 O15379 1/20 0.38
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
POLB P06746 2/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TRPM8 Q7Z2W7 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
PARP1 P09874 1/20 0.33
GPR6 P46095 1/20 0.33
MAPT P10636 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1684122 0.78 RIPK1 (0.43) RIPK1TRPM8GABRA1GABRG2GABRB3
SCHEMBL1684143 0.76 RIPK1 (0.42) RIPK1KDM4EALDH1A1GABRA1GABRG2
SCHEMBL1684139 0.72 TDO2 (0.40) RIPK1TRPM8RAB9A
SCHEMBL1684181 0.72 MPO (0.42)
SCHEMBL1684118 0.70 TDO2 (0.36) RIPK1HDAC3POLBTRPM8
SCHEMBL1684177 0.68 RIPK1 (0.45) RIPK1TRPM8
SCHEMBL40939 0.66 KDM4E (0.49) CTNNB1WNT3AHTTSMN1; SMN2KDM4E
SCHEMBL2234661 0.65 KDM4E (0.44) CTNNB1WNT3AHTTSMN1; SMN2KDM4E
SCHEMBL15078308 0.65 KDM4E (0.44) CTNNB1WNT3APOLBHTTSMN1; SMN2
SCHEMBL4783535 0.64 TRPM8 (0.55) RIPK1HDAC3TRPM8RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011041512-A2 COMPOSITIONS AND METHODS FOR TREATING MLV-INFECTION, AND PREVENTING AND TREATING MLV-INITIATED DISEASES EMORY UNIVERSITY (US) 2011-04-07 WO disclosed