SCHEMBL16974396

SCHEMBL16974396

C=CC(=O)N(c1cc(Br)ccc1Br)C(O)C#N

nearest known ligand 0.31

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.31
KMT2A Q03164 3/20 0.31
MEN1 O00255 2/20 0.31
LMNA P02545 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
THRB P10828 1/20 0.31
BLM P54132 1/20 0.31
BTK Q06187 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PLK3 Q9H4B4 1/20 0.31
TGM2 P21980 2/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16167178 0.72 SIGMAR1 (0.41) ALDH1A1LMNABTKNPSR1TGM2
SCHEMBL16095632 0.65 EGFR (0.39) ALDH1A1LMNABTKTGM2CYP2C19
SCHEMBL31289612 0.64 MAPK3 (0.37) ALDH1A1KMT2AMEN1LMNAGAA
SCHEMBL4654542 0.63 ALDH1A1 (0.39) ALDH1A1KMT2AMEN1LMNACYP1A2
SCHEMBL11428595 0.58 FAAH (0.30)
SCHEMBL19643823 0.57 MEN1 (0.54) ALDH1A1KMT2AMEN1LMNACYP1A2
SCHEMBL3663002 0.57 DGAT1 (0.38) ALDH1A1LMNACYP1A2CYP2C9ALOX15
SCHEMBL16684492 0.57 HPGD (0.33) ALDH1A1KMT2AMEN1LMNACYP3A4
SCHEMBL2787330 0.55 HSP90AA1 (0.41) ALDH1A1LMNAALOX15TSHR
SCHEMBL9485990 0.55 CCR5 (0.42) ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3099309-A1 CHEMOTHERAPEUTIC DRUG COMBINATION Yeditepe Universitesi (TR) 2016-12-07 EP disclosed
WO-2015116012-A1 CHEMOTHERAPEUTIC DRUG COMBINATION YEDITEPE UNIVERSITESI (TR) 2015-08-06 WO disclosed