SCHEMBL17023484

SCHEMBL17023484

CC(=O)c1cn(CC(=O)O)c2ccc(O)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
CREBBP Q92793 3/20 0.49
SMN1; SMN2 Q16637 5/20 0.48
ALDH1A1 P00352 4/20 0.48
LMNA P02545 3/20 0.48
KDM4E B2RXH2 3/20 0.48
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
MAPT P10636 2/20 0.45
KAT2B Q92831 1/20 0.44
CNR2 P34972 2/20 0.43
CNR1 P21554 1/20 0.43
RXFP1 Q9HBX9 2/20 0.43
HTT P42858 2/20 0.42
CFD P00746 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
STAT3 P40763 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17023330 0.88 KMT2A (0.49) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL23704991 0.88 KMT2A (0.49) KMT2AALDH1A1KDM4EMAPTCNR2
SCHEMBL18549503 0.85 KMT2A (0.47) KMT2AALDH1A1KDM4EMAPTCNR2
SCHEMBL25925010 0.85 SMN1; SMN2 (0.53) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL17038773 0.85 GAA (0.54) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL17023688 0.84 CFD (0.49) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL29781757 0.84 CFD (0.49) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL12480373 0.82 ALDH1A1 (0.56) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL18554040 0.82 PTGDR2 (0.47) KMT2ACREBBPSMN1; SMN2ALDH1A1LMNA
SCHEMBL12479682 0.81 HTR6 (0.43) CREBBPSMN1; SMN2ALDH1A1LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 102 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10689409-B2 Amino compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-06-23 US disclosed
US-10689409-B2 Amino compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-06-23 US disclosed
US-10660876-B2 Amino compounds for treatment of medical disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-05-26 US disclosed
US-10660876-B2 Amino compounds for treatment of medical disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-05-26 US disclosed
US-10550140-B2 Ether compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-02-04 US disclosed
US-10550140-B2 Ether compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2020-02-04 US disclosed
US-10428094-B2 Amide compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2019-10-01 US disclosed
US-10428094-B2 Amide compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2019-10-01 US disclosed
US-10385097-B2 Ether compounds for treatment of medical disorders ACHILLION PHARMACEUTICALS, INC. (US) 2019-08-20 US disclosed
US-10385097-B2 Ether compounds for treatment of medical disorders ACHILLION PHARMACEUTICALS, INC. (US) 2019-08-20 US disclosed
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239893-A1 Amide Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239893-A1 Amide Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239837-A1 Factor D Inhibitors Useful for Treating Inflammatory Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239893-A1 Amide Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239837-A1 Factor D Inhibitors Useful for Treating Inflammatory Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239837-A1 Factor D Inhibitors Useful for Treating Inflammatory Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150239919-A1 Carbamate, Ester, and Ketone Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
US-20150166641-A1 Compositions and Methods for the Removal of Biofilms UNIV SOUTHERN CALIFORNIA (US) 2015-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10550140-B2 Ether compounds for treatment of complement mediated disorders TFPI, CFD, C9 KMT2A 3926/4885CREBBP 1802/4885SMN1; SMN2 890/4885
US-10385097-B2 Ether compounds for treatment of medical disorders CFD, TFPI, F12 KMT2A 3998/4885CREBBP 1184/4885SMN1; SMN2 2749/4885
US-20150239837-A1 Factor D Inhibitors Useful for Treating Inflammatory Disorders CFD, TFPI, TFPI2 KMT2A 4720/4885CREBBP 2125/4885SMN1; SMN2 2680/4885
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders CFD, TFPI, C9 KMT2A 4197/4885CREBBP 2836/4885SMN1; SMN2 1331/4885
US-10660876-B2 Amino compounds for treatment of medical disorders CFD, CFH, F12 KMT2A 4309/4885CREBBP 3434/4885SMN1; SMN2 1899/4885
US-10428094-B2 Amide compounds for treatment of complement mediated disorders CFD, TFPI, C9 KMT2A 4064/4885CREBBP 1853/4885SMN1; SMN2 1358/4885
US-20150166641-A1 Compositions and Methods for the Removal of Biofilms FCGR3B, FGB, CD47 KMT2A 4429/4885CREBBP 3692/4885SMN1; SMN2 4777/4885
US-20150239893-A1 Amide Compounds for Treatment of Complement Mediated Disorders CFD, TFPI, C9 KMT2A 4064/4885CREBBP 1853/4885SMN1; SMN2 1358/4885
US-10689409-B2 Amino compounds for treatment of complement mediated disorders CFD, TFPI, C9 KMT2A 4197/4885CREBBP 2836/4885SMN1; SMN2 1331/4885
US-20150239919-A1 Carbamate, Ester, and Ketone Compounds for Treatment of Complement Mediated Disorders CFD, C9, CFH KMT2A 2789/4885CREBBP 724/4885SMN1; SMN2 2371/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.