SCHEMBL17039280

SCHEMBL17039280

Cc1cn2cc(-c3cccc(-c4ccccc4F)c3)nc2c(-c2ccccc2F)c1CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.44
LMNA P02545 1/20 0.44
PDCD1 Q15116 3/20 0.39
CD274 Q9NZQ7 3/20 0.39
CTSA P10619 2/20 0.38
KDM4E B2RXH2 5/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
ALDH1A1 P00352 4/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
GRIN2B Q13224 1/20 0.36
TMIGD3 P0DMS9 2/20 0.36
LTB4R Q15722 1/20 0.36
SCN9A Q15858 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17039278 0.83 FABP4 (0.41) SMN1; SMN2LMNA
SCHEMBL17039277 0.80 NR1I2 (0.42) SMN1; SMN2LMNAPDCD1CD274KDM4E
SCHEMBL17029051 0.78 NR1I2 (0.39) SCN9A
SCHEMBL17039256 0.75 NR1I2 (0.41) PDCD1CD274KDM4ERAB9ANPC1
SCHEMBL20344804 0.73 ALDH1A3 (0.34) SMN1; SMN2PDCD1CD274RAB9ANPC1
SCHEMBL20344807 0.73 P2RX7 (0.33)
SCHEMBL20344808 0.71 GNRHR (0.35) SMN1; SMN2KDM4ERAB9ANPC1ALDH1A1
SCHEMBL3802345 0.64 LMNA (0.48) SMN1; SMN2LMNAKDM4ERAB9AALDH1A1
SCHEMBL9890675 0.62 SMN1; SMN2 (0.49) SMN1; SMN2LMNAKDM4E
SCHEMBL12856837 0.61 PTPRC (0.55) SMN1; SMN2RAB9ANPC1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015126765-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-08-27 WO disclosed