SCHEMBL17065417

SCHEMBL17065417

COC(=O)N[C@@H](Cc1ccc(-c2ccncc2)cc1)C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.44
ITGB7 P26010 2/20 0.44
ROCK2 O75116 5/20 0.43
ROCK1 Q13464 5/20 0.43
PRKACA P17612 3/20 0.43
IRAK1 P51617 3/20 0.43
PRKG1 Q13976 3/20 0.43
PKN2 Q16513 3/20 0.43
CLK4 Q9HAZ1 3/20 0.43
PRKX P51817 2/20 0.43
RPS6KB1 P23443 2/20 0.43
PRKG2 Q13237 2/20 0.43
HIPK4 Q8NE63 2/20 0.43
AURKB Q96GD4 2/20 0.43
LIMK1 P53667 1/20 0.43
CSNK1G1 Q9HCP0 1/20 0.43
MME P08473 2/20 0.42
HPGDS O60760 2/20 0.42
ACACB O00763 1/20 0.42
RPS6KA5 O75582 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16823433 0.87 HPGDS (0.53) MMEHPGDSCTSSCTSK
SCHEMBL2714739 0.87 CTSS (0.56) ITGA4ITGB7CYP17A1LHCGRCTSS
SCHEMBL2714740 0.87 CTSS (0.56) ITGA4ITGB7CYP17A1LHCGRCTSS
SCHEMBL14850462 0.81 ACACB (0.46) ITGA4ITGB7ROCK2ROCK1ACACB
SCHEMBL20241397 0.80 LDHA (0.53) ACACB
SCHEMBL20241398 0.80 LDHA (0.53) ACACB
SCHEMBL3616169 0.80 MMP1 (0.55) HPGDSALDH1A1HSD17B10CTSSCTSK
SCHEMBL3616167 0.80 MMP1 (0.55) HPGDSALDH1A1HSD17B10CTSSCTSK
SCHEMBL15577717 0.80 NOS3 (0.49) MMECTSK
SCHEMBL4516299 0.79 GPR142 (0.50) ITGA4ROCK2ROCK1PRKACAIRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3113780-A1 HIV PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-01-11 EP claimed
WO-2015134366-A1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-09-11 WO claimed