SCHEMBL1708680

SCHEMBL1708680

CCOc1nc2ccc(OC)cc2n1-c1cccc(CNc2ccc3c(c2)OC[C@H]3OC(C)=O)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.39
MTNR1B P49286 7/20 0.39
MAPT P10636 5/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
CLK1 P49759 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ACACB O00763 1/20 0.33
FFAR1 O14842 2/20 0.33
PDE2A O00408 1/20 0.33
CD274 Q9NZQ7 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
TP53 P04637 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708014 0.91 MAPT (0.35) MAPTALDH1A1HTTNPSR1FFAR1
SCHEMBL1708303 0.91 SMN1; SMN2 (0.37) MAPTALDH1A1HTTCLK1NPSR1
SCHEMBL10291805 0.89 MTNR1A (0.39) MTNR1AMTNR1BMAPTALDH1A1HTT
SCHEMBL10292315 0.89 MTNR1A (0.39) MTNR1AMTNR1BMAPTALDH1A1HTT
SCHEMBL1708151 0.88 FFAR1 (0.40) MTNR1AMTNR1BMAPTFFAR1NPC1
SCHEMBL1708678 0.88 FFAR1 (0.46) MTNR1AMTNR1BFFAR1
SCHEMBL1708622 0.86 TSHR (0.35) MAPTALDH1A1HTTNPSR1CD274
SCHEMBL1708148 0.86 MTNR1A (0.41) MTNR1AMTNR1BMAPTALDH1A1HTT
SCHEMBL1708693 0.85 SMN1; SMN2 (0.36) MAPTALDH1A1HTTCLK1NPSR1
SCHEMBL1707875 0.83 HPGD (0.37) MAPTALDH1A1NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed