SCHEMBL17090273

SCHEMBL17090273

Cc1c(C)c(C(=O)NC(C)C)c(C)c(C)c1NCCCCCNS(=O)(=O)C(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.32
GRIA1 P42261 3/20 0.30
TAS1R3 Q7RTX0 3/20 0.30
TAS1R1 Q7RTX1 3/20 0.30
TAS1R2 Q8TE23 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090288 0.85 GRIA1 (0.49) EPHX1GRIA1
SCHEMBL10115148 0.85 ALDH1A1 (0.38)
SCHEMBL17090272 0.83 ALDH1A1 (0.32)
SCHEMBL11935695 0.79 PAOX (0.37) EPHX1TAS1R3TAS1R1TAS1R2
SCHEMBL17090276 0.76 CISD1 (0.34)
SCHEMBL11935627 0.76 LMNA (0.36)
SCHEMBL13565343 0.76 MLYCD (0.45)
SCHEMBL11935634 0.74 TAS1R3 (0.37) TAS1R3TAS1R1
SCHEMBL11935350 0.74 BRD4 (0.38) TAS1R3TAS1R1
SCHEMBL11935606 0.72 NPSR1 (0.46) TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed