SCHEMBL17090287

SCHEMBL17090287

Cc1cc(NCCCCCNS(=O)(=O)C(C)C)c(C)c(C(=O)NC(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 3/20 0.43
NPY5R Q15761 6/20 0.39
NR3C1 P04150 2/20 0.39
CISD1 Q9NZ45 5/20 0.33
FABP4 P15090 1/20 0.33
HTR1A P08908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090276 0.87 CISD1 (0.34) NR3C1CISD1FABP4
SCHEMBL10115460 0.86 ALDH1A1 (0.39) GRIA1NR3C1FABP4
SCHEMBL13564980 0.84 GRIA1 (0.43) GRIA1NPY5RHTR1A
SCHEMBL11935696 0.83 ROCK1 (0.41)
SCHEMBL13439365 0.82 GRIA1 (0.43) GRIA1NPY5RCISD1FABP4HTR1A
SCHEMBL17090215 0.78 GRIA1 (0.44) GRIA1NPY5RNR3C1FABP4HTR1A
SCHEMBL17090450 0.77 GRIA1 (0.43) GRIA1NPY5RNR3C1
SCHEMBL17090288 0.75 GRIA1 (0.49) GRIA1NPY5RFABP4HTR1A
SCHEMBL17090505 0.75 NR3C1 (0.39) NR3C1
SCHEMBL17090544 0.73 MAPK14 (0.37) NPY5RNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed