SCHEMBL1709238

SCHEMBL1709238

CC(NCC1CC12CCN(c1ccccc1)CC2)c1ccc(F)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.59
RAD52 P43351 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
MAPT P10636 2/20 0.40
MITF O75030 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
MC4R P32245 1/20 0.39
CCR3 P51677 2/20 0.39
ATM Q13315 1/20 0.37
NPY1R P25929 1/20 0.37
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
HTR1A P08908 2/20 0.36
HTR7 P34969 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709240 0.75 SCN9A (0.60) SCN9AALDH1A1KMT2ACCR3ATM
SCHEMBL17389438 0.75 SCN9A (0.48) SCN9ALMNA
SCHEMBL20567442 0.75 SCN9A (0.48) SCN9ALMNA
SCHEMBL1709252 0.75 SCN9A (0.56) SCN9ALMNAKMT2ASIGMAR1
SCHEMBL1709236 0.74 SCN9A (1.00) SCN9AMAPTALDH1A1HTTKMT2A
SCHEMBL1709241 0.72 SCN9A (0.54) SCN9AALDH1A1NPY1RHTR7SIGMAR1
SCHEMBL10072038 0.70 SCN9A (0.53) SCN9AALDH1A1LMNAKMT2AHTR7
SCHEMBL18298019 0.70 NAMPT (0.55) ATM
SCHEMBL1709243 0.69 SCN9A (0.52) SCN9AMAPTLMNAKMT2APOLB
SCHEMBL1709237 0.67 SCN9A (0.58) SCN9AHTR1ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed