SCHEMBL1709236

SCHEMBL1709236

c1ccc(CC(NCC2CC23CCN(c2ccccc2)CC3)c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 1.00
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 2/20 0.36
GFER P55789 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
DRD4 P21917 1/20 0.35
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 2/20 0.34
NAMPT P43490 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
USP2 O75604 1/20 0.33
CYP2D6 P10635 1/20 0.33
NCOA1 Q15788 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709240 0.75 SCN9A (0.60) SCN9AL3MBTL1GFERSIGMAR1ALDH1A1
SCHEMBL1709238 0.74 SCN9A (0.59) SCN9AMAPTPOLBSIGMAR1ALDH1A1
SCHEMBL1709252 0.72 SCN9A (0.56) SCN9ASIGMAR1MEN1KMT2ADRD2
SCHEMBL1709241 0.71 SCN9A (0.54) SCN9AL3MBTL1GFERSIGMAR1ALDH1A1
SCHEMBL1709251 0.70 SCN9A (0.54) SCN9AMAPTGFERALDH1A1KDM4E
SCHEMBL10072038 0.69 SCN9A (0.53) SCN9AALDH1A1MEN1KMT2AUSP2
SCHEMBL1709249 0.69 DRD4 (0.60) SCN9ASIGMAR1DRD4ALDH1A1KDM4E
SCHEMBL1709243 0.68 SCN9A (0.52) SCN9AMAPTPOLBKDM4EMEN1
SCHEMBL1286796 0.67 USP2 (0.49) SCN9AL3MBTL1POLBSIGMAR1ALDH1A1
SCHEMBL10071960 0.66 SCN9A (0.49) SCN9AMAPTALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed