SCHEMBL1709252

SCHEMBL1709252

CCCCCC(C)NCC1CC12CCN(c1ccccc1)CC2

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.56
DPP4 P27487 2/20 0.39
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
LMNA P02545 1/20 0.35
PLA2G1B P04054 1/20 0.35
TSHR P16473 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
DRD2 P14416 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
OPRM1 P35372 3/20 0.34
OPRD1 P41143 3/20 0.34
OPRK1 P41145 3/20 0.34
OPRL1 P41146 3/20 0.34
CHRNA7 P36544 1/20 0.34
GRM2 Q14416 4/20 0.34
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709238 0.75 SCN9A (0.59) SCN9AKMT2ALMNASIGMAR1
SCHEMBL1709241 0.75 SCN9A (0.54) SCN9ADPP4DRD2SIGMAR1CHRNA7
SCHEMBL1709240 0.73 SCN9A (0.60) SCN9AKMT2ASIGMAR1MEN1
SCHEMBL1709236 0.72 SCN9A (1.00) SCN9AKMT2ADRD2SIGMAR1MEN1
SCHEMBL10072038 0.70 SCN9A (0.53) SCN9AKMT2ALMNATSHRCHRNA7
SCHEMBL1709243 0.69 SCN9A (0.52) SCN9AKMT2ALMNAMEN1
SCHEMBL1709237 0.69 SCN9A (0.58) SCN9ADRD2SIGMAR1
SCHEMBL1709251 0.66 SCN9A (0.54) SCN9AKMT2AMEN1
SCHEMBL1709217 0.66 SCN9A (0.48) SCN9AKMT2ALMNATSHR
SCHEMBL11668124 0.66 DRD2 (0.49) KMT2ANPSR1LMNAPLA2G1BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed