SCHEMBL1709413

SCHEMBL1709413

C=C(O)C[C@@H]1CC[C@@H](N(CC2CCCCC2)CC2CCCCC2)[C@H](c2cccc(Cl)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 16/20 0.41
TP53 P04637 11/20 0.41
EPHX2 P34913 1/20 0.37
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
SLC9A1 P19634 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033115 0.82 MDM2 (0.43) MDM2TP53EPHX2
SCHEMBL1709502 0.81 ESR2 (0.35)
SCHEMBL1709411 0.80 SIGMAR1 (0.31)
SCHEMBL10033138 0.80 SIGMAR1 (0.42) HTR2AHTR2CHTR2B
SCHEMBL10033140 0.79 OPRM1 (0.32) HTR2CHTR2B
SCHEMBL1709403 0.77 HTR2C (0.34) TP53HTR2AHTR2C
SCHEMBL1709404 0.77 HTR2C (0.34) TP53HTR2AHTR2C
SCHEMBL1709443 0.77 HTR2C (0.34) TP53HTR2AHTR2C
SCHEMBL10032995 0.77 HTR2A (0.34) HTR2AHTR2CHTR2B
SCHEMBL1709491 0.77 KDM1A (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed