SCHEMBL1709491

SCHEMBL1709491

C=C(O)C[C@@H]1CC[C@@H](N(CCC2CCCCC2)CCC2CCCCC2)[C@H](c2ccccc2)C1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.42
MAOB P27338 5/20 0.42
MAOA P21397 3/20 0.42
GPR88 Q9GZN0 3/20 0.39
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709420 0.90 SIGMAR1 (0.40) KDM1AMAOBMAOAGPR88SIGMAR1
SCHEMBL10032995 0.88 HTR2A (0.34) KDM1AMAOBMAOABCHEACHE
SCHEMBL1709402 0.88 HTR2C (0.34) KDM1AMAOBMAOASIGMAR1
SCHEMBL10032988 0.87 KDM1A (0.33) KDM1AMAOBMAOABCHE
SCHEMBL1709423 0.85 ACHE (0.30) KDM1AMAOBMAOAACHE
SCHEMBL10033139 0.85 SIGMAR1 (0.39) KDM1AMAOBMAOASIGMAR1
SCHEMBL1709450 0.83 HTR2C (0.33) KDM1AMAOBMAOA
SCHEMBL10032822 0.83 HTR2C (0.33) KDM1AMAOBMAOA
SCHEMBL1709412 0.81 OPRM1 (0.31) KDM1AMAOBMAOABCHEACHE
SCHEMBL10033004 0.80 PSEN1 (0.36) GPR88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed