SCHEMBL1709420

SCHEMBL1709420

C=C(O)C[C@@H]1CC[C@@H](N(CCC2CCCCC2)CCC2CCCCC2)[C@H](c2ccc(F)cc2)C1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.40
KDM1A O60341 5/20 0.33
MAOA P21397 4/20 0.33
MAOB P27338 4/20 0.33
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GPR88 Q9GZN0 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
SLC6A2 P23975 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
HTR2B P41595 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033139 0.95 SIGMAR1 (0.39) SIGMAR1KDM1AMAOAMAOBPOLB
SCHEMBL1709491 0.90 KDM1A (0.42) SIGMAR1KDM1AMAOAMAOBGPR88
SCHEMBL1709402 0.89 HTR2C (0.34) SIGMAR1KDM1AMAOAMAOBSMN1; SMN2
SCHEMBL10033138 0.89 SIGMAR1 (0.42) SIGMAR1KDM1APOLBRAB9ASMN1; SMN2
SCHEMBL10032995 0.87 HTR2A (0.34) KDM1AMAOAMAOBHTR2AHTR2C
SCHEMBL10032988 0.86 KDM1A (0.33) KDM1AMAOAMAOB
SCHEMBL1709423 0.84 ACHE (0.30) KDM1AMAOAMAOB
SCHEMBL10032822 0.84 HTR2C (0.33) KDM1AMAOAMAOBHTR2AHTR2C
SCHEMBL1709450 0.84 HTR2C (0.33) KDM1AMAOAMAOBHTR2AHTR2C
SCHEMBL10033004 0.81 PSEN1 (0.36) GPR88SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed