SCHEMBL17100575

SCHEMBL17100575

CC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCN

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 8/20 1.00
HIF1A Q16665 1/20 1.00
TET2 Q6N021 1/20 1.00
DOHH Q9BU89 1/20 1.00
KDM4E B2RXH2 1/20 0.92
LMNA P02545 1/20 0.92
GAA P10253 1/20 0.92
SMN1; SMN2 Q16637 1/20 0.92
PAOX Q6QHF9 3/20 0.46
SLC6A5 Q9Y345 2/20 0.44
KDM4C Q9H3R0 7/20 0.40
CASP2 P42575 1/20 0.38
KDM5A P29375 1/20 0.37
KDM7A Q6ZMT4 1/20 0.37
PHF8 Q9UPP1 1/20 0.37
KDM2A Q9Y2K7 1/20 0.37
NAAA Q02083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17109729 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
SCHEMBL13367139 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
SCHEMBL21051754 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
Deferoxamine SCHEMBL10498260 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
Deferoxamine SCHEMBL34571 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
SCHEMBL19040665 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
SCHEMBL26511991 1.00 KDM4A (1.00) KDM4AHIF1ATET2DOHHKDM4E
Deferoxamine SCHEMBL20658962 0.99 KDM4A (0.97) KDM4AHIF1ATET2DOHHKDM4E
Deferoxamine SCHEMBL21049242 0.99 KDM4A (0.97) KDM4AHIF1ATET2DOHHKDM4E
Deferoxamine SCHEMBL20658960 0.99 KDM4A (0.97) KDM4AHIF1ATET2DOHHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025088147-A1 THERANOSTIC PSMA-TARGETING LIGANDS FOR THE DIAGNOSIS AND TREATMENT OF PSMA-EXPRESSING CANCERS AND THEIR SOLID PHASE SYNTHESIS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2025-05-01 WO claimed
US-20230406847-A1 LIGANDS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) CONTAINING HETEROAROMATIC LINKER BUILDING BLOCKS ABX ADVANCED BIOCHEMICAL COMPOUNDS GMBH (DE) 2023-12-21 US claimed
EP-4244216-A1 LIGANDS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) CONTAINING HETEROAROMATIC LINKER BUILDING BLOCKS ABX Advanced Biochemical Compounds GmbH (DE) 2023-09-20 EP claimed
WO-2022101352-A1 LIGANDS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) CONTAINING HETEROAROMATIC LINKER BUILDING BLOCKS ABX ADVANCED BIOCHEMICAL COMPOUNDS GMBH (DE) 2022-05-19 WO claimed
EP-4577578-A1 DLL3 BINDING MOLECULES AND USES THEREOF Abdera Therapeutics Inc. (US) 2025-07-02 EP disclosed
EP-4577526-A1 VHH ANTIBODY CONJUGATES Abdera Therapeutics Inc. (US) 2025-07-02 EP disclosed
EP-4577250-A1 MULTIVALENT IMMUNOCONJUGATES FOR TARGETED RADIOISOTOPE THERAPY Abdera Therapeutics Inc. (US) 2025-07-02 EP disclosed
WO-2025088147-A1 THERANOSTIC PSMA-TARGETING LIGANDS FOR THE DIAGNOSIS AND TREATMENT OF PSMA-EXPRESSING CANCERS AND THEIR SOLID PHASE SYNTHESIS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2025-05-01 WO disclosed
US-20250127938-A1 THERAGNOSTIC FOLATE CONJUGATES MERCK PATENT GMBH (DE) 2025-04-24 US disclosed
US-20250108138-A1 THERAGNOSTIC FOLATE CONJUGATES MERCK PATENT GMBH (DE) 2025-04-03 US disclosed
EP-4472677-A1 THERAGNOSTIC FOLATE CONJUGATES Merck Patent GmbH (DE) 2024-12-11 EP disclosed
EP-4472676-A1 THERAGNOSTIC FOLATE CONJUGATES Merck Patent GmbH (DE) 2024-12-11 EP disclosed
EP-3131585-B1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY UNIV ZUERICH (CH) 2020-07-15 EP disclosed
EP-3131585-B1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY UNIV ZUERICH (CH) 2020-07-15 EP disclosed
US-20170106106-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY UNIVERSITAT ZURICH (CH) 2017-04-20 US disclosed
US-20170106106-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY UNIVERSITAT ZURICH (CH) 2017-04-20 US disclosed
US-20170106106-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY UNIVERSITAT ZURICH (CH) 2017-04-20 US disclosed
EP-3131585-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY Universität Zürich (CH) 2017-02-22 EP disclosed
WO-2015140212-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY Universität Zürich (CH) 2015-09-24 WO disclosed
WO-2015140212-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY Universität Zürich (CH) 2015-09-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170106106-A1 MULTIDENTATE BIFUNCTIONAL CHELATING AGENTS FOR RADIONUCLIDE COMPLEXATION IN DIAGNOSTICS AND THERAPY AOC1, XDH, FOLR1 KDM4A 3400/4885HIF1A 1613/4885TET2 4608/4885
US-20230406847-A1 LIGANDS OF PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) CONTAINING HETEROAROMATIC LINKER BUILDING BLOCKS KLK3, FOLH1, BPHL KDM4A 1803/4885HIF1A 1645/4885TET2 4858/4885
US-20250108138-A1 THERAGNOSTIC FOLATE CONJUGATES FOLR1, MTHFD1, MTHFD2 KDM4A 2724/4885HIF1A 2958/4885TET2 361/4885
US-20250127938-A1 THERAGNOSTIC FOLATE CONJUGATES FOLR1, FOLR2, DHFR KDM4A 2949/4885HIF1A 4050/4885TET2 544/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.