SCHEMBL17184754

SCHEMBL17184754

NNC(=O)c1ccc(I)cc1C(=O)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
GFER P55789 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
MAP2K1 Q02750 3/20 0.36
RAF1 P04049 1/20 0.36
PDGFRB P09619 1/20 0.36
CSNK2A2 P19784 1/20 0.36
MAP2K2 P36507 1/20 0.36
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36
CSNK2A3 Q8NEV1 1/20 0.36
AURKC Q9UQB9 1/20 0.36
CAMK2A Q9UQM7 1/20 0.36
MEN1 O00255 1/20 0.35
MITF O75030 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
NCOA1 Q15788 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11382111 0.78 CTSD (0.47) ALDH1A1GFERMAPTKDM4EMEN1
SCHEMBL17185444 0.77 ALDH1A1 (0.44) ALDH1A1GFERMAPTKDM4EMEN1
SCHEMBL1974542 0.74 ALDH1A1 (0.48) ALDH1A1GFERMAPTKDM4EMAP2K1
SCHEMBL2721634 0.73 MAPT (0.53) ALDH1A1GFERMAPTKDM4EMEN1
SCHEMBL15471934 0.71 KDM4E (0.44) ALDH1A1GFERMAPTKDM4EMAP2K1
SCHEMBL15471931 0.71 ALDH1A1 (0.44) ALDH1A1GFERMAPTKDM4EMAP2K1
SCHEMBL15471933 0.71 ALDH1A1 (0.68) ALDH1A1GFERMAPTKDM4EMEN1
SCHEMBL16192428 0.64 ALDH1A1 (0.53) ALDH1A1GFERMAPTKDM4EMEN1
SCHEMBL8272560 0.64 SIRT2 (0.42) ALDH1A1MAPTKDM4EMEN1MITF
SCHEMBL27775502 0.64 MGLL (0.48) MEN1GAAKMT2ANPSR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161014-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed