SCHEMBL17185444

SCHEMBL17185444

CC(=O)c1cc(I)ccc1C(=O)NN

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
GFER P55789 2/20 0.44
MAPT P10636 5/20 0.43
KDM4E B2RXH2 4/20 0.43
GAA P10253 3/20 0.39
CTSD P07339 2/20 0.39
MEN1 O00255 1/20 0.39
MITF O75030 1/20 0.39
KMT2A Q03164 1/20 0.39
NCOA1 Q15788 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
P2RX7 Q99572 1/20 0.38
PTPRC P08575 1/20 0.37
PTPN2 P17706 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPRA P18433 1/20 0.37
PTPRB P23467 1/20 0.37
PTPRE P23469 1/20 0.37
PTPN6 P29350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21592065 0.82 PTPRC (0.40) ALDH1A1MAPTKDM4EGAAMEN1
SCHEMBL15471934 0.80 KDM4E (0.44) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL1974542 0.79 ALDH1A1 (0.48) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL2721634 0.78 MAPT (0.53) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL21592068 0.77 PTPRC (0.49) ALDH1A1KDM4EPTPRCPTPN2PTPN1
SCHEMBL17184754 0.77 ALDH1A1 (0.40) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL15471931 0.76 ALDH1A1 (0.44) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL15471933 0.76 ALDH1A1 (0.68) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL8219059 0.75 CTSD (0.58) ALDH1A1GFERMAPTKDM4EGAA
SCHEMBL9117052 0.73 PTPRC (0.49) ALDH1A1KDM4EPTPRCPTPN2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161011-A1 BENZAMIDE CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed