SCHEMBL1720288

SCHEMBL1720288

CC(C)N(C(=O)c1nc(N2CCNCC2)nc2sc(-c3ccc(F)cc3)cc12)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 1/20 0.39
USP28 Q96RU2 1/20 0.38
USP25 Q9UHP3 1/20 0.38
HRH4 Q9H3N8 2/20 0.37
HDAC3 O15379 4/20 0.36
HDAC2 Q92769 3/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
SCN9A Q15858 2/20 0.35
HDAC1 Q13547 1/20 0.35
KIT P10721 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
MAPK14 Q16539 1/20 0.34
CNR2 P34972 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793765 0.71 ALDH1A1 (0.45) HDAC3HTR1AHTR7USP2ALDH1A1
SCHEMBL1720286 0.70 FPR2 (0.37) HDAC3HDAC2SCN9AKITCYP1A2
SCHEMBL655170 0.70 CNR2 (0.48) HRH4KITCNR2ALDH1A1TSHR
SCHEMBL655042 0.69 HRH4 (0.61) HRH4HRH3CNR2ALDH1A1TSHR
SCHEMBL4560186 0.62 HDAC1 (0.43) HRH4HDAC3HDAC2SCN9AHDAC1
SCHEMBL4560538 0.61 MKNK2 (0.46) SCN9AHDAC1USP2ALDH1A1CYP1A2
SCHEMBL11201732 0.60 P2RY12 (0.48) P2RY12HRH4ALDH1A1TSHRCASP1
SCHEMBL654538 0.59 ALDH1A1 (0.75) ALDH1A1
SCHEMBL655041 0.59 USP2 (0.35) HRH4HDAC3HDAC2HTR1AHTR7
SCHEMBL798319 0.59 CHEK1 (0.46) HTR1AHTR7USP2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2405973-A2 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-01-18 EP disclosed
WO-2010103130-A2 NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-09-16 WO disclosed