SCHEMBL172307

SCHEMBL172307

CC[C@H](C)CNCc1ccc2c(c1)OC[C@@H]1C[C@@H]21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
MCHR1 Q99705 1/20 0.32
KMT2A Q03164 3/20 0.32
LTA4H P09960 2/20 0.32
MEN1 O00255 2/20 0.32
BDKRB1 P46663 1/20 0.31
HPGD P15428 1/20 0.31
LTB4R Q15722 1/20 0.30
LTB4R2 Q9NPC1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4145157 0.76 ALDH1A1 (0.41) ALDH1A1KDM4ETSHRMCHR1KMT2A
SCHEMBL6869567 0.67 CYP19A1 (0.39) ALDH1A1DRD2DRD3
SCHEMBL21799751 0.65 ANPEP (0.50) ALDH1A1
SCHEMBL4152298 0.65 OPRD1 (0.40) BDKRB1
SCHEMBL172730 0.65 DNM1 (0.49) ALDH1A1KDM4EHPGD
SCHEMBL14847248 0.64 KDM4E (0.56) ALDH1A1KDM4ETSHRMCHR1KMT2A
SCHEMBL13039461 0.64 ALDH1A1 (0.59) ALDH1A1KDM4ETSHRKMT2AMEN1
SCHEMBL14847238 0.64 ALDH1A1 (0.59) ALDH1A1KDM4ETSHRKMT2AMEN1
SCHEMBL38653550 0.64 DRD2 (0.57) ALDH1A1DRD2DRD3KMT2AMEN1
SCHEMBL21799963 0.64 ADRB2 (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed