SCHEMBL172552

SCHEMBL172552

CCC[C@H](NC)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
AOC3 Q16853 2/20 0.47
HTR2A P28223 3/20 0.47
HRH1 P35367 2/20 0.47
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
CHRM2 P08172 2/20 0.41
ADRA1A P35348 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
RGS12 O14924 1/20 0.41
GLA P06280 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
ALOX12 P18054 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL172587 1.00 ALDH1A1 (0.49) ALDH1A1AOC3HTR2AHRH1MAPT
SCHEMBL13075028 1.00 ALDH1A1 (0.49) ALDH1A1AOC3HTR2AHRH1MAPT
SCHEMBL4591305 0.89 LMNA (0.50) ALDH1A1AOC3HTR2AHRH1MAPT
SCHEMBL14533617 0.88 POLB (0.46) ALDH1A1AOC3HTR2AHRH1MAPT
SCHEMBL14533565 0.86 ALDH1A1 (0.45) ALDH1A1HTR2AHRH1MAPTTACR3
SCHEMBL11638197 0.84 AOC3 (0.48) ALDH1A1AOC3HTR2AHRH1MAPT
SCHEMBL11256309 0.84 TACR3 (0.44) ALDH1A1HTR2AHRH1TACR3
SCHEMBL9149427 0.84 TACR3 (0.44) ALDH1A1HTR2AHRH1TACR3
SCHEMBL11153215 0.84 TACR3 (0.44) ALDH1A1HTR2AHRH1TACR3
SCHEMBL8695928 0.84 LTA4H (0.47) ALDH1A1MAPTHTTTSHRALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8288569-B2 Carbonyl asymmetric alkylation SANDOZ AG (CH) 2012-10-16 US disclosed
US-8288569-B2 Carbonyl asymmetric alkylation SANDOZ AG (CH) 2012-10-16 US disclosed
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed
EP-1966127-B1 CARBONYL ASYMMETRIC ALKYLATION SANDOZ AG (CH) 2011-04-06 EP disclosed
US-20110009648-A1 Carbonyl Asymmetric Alkylation SANDOZ AG (CH) 2011-01-13 US disclosed
US-20110009648-A1 Carbonyl Asymmetric Alkylation SANDOZ AG (CH) 2011-01-13 US disclosed
WO-2007082771-A1 CARBONYL ASYMMETRIC ALKYLATION SANDOZ AG (CH) 2007-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110009648-A1 Carbonyl Asymmetric Alkylation COASY, ADH5, SI ALDH1A1 53/4885AOC3 345/4885HTR2A 496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.