SCHEMBL17347402

SCHEMBL17347402

COCCNC(=O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.61
MAOA P21397 2/20 0.61
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
TCF4 P15884 2/20 0.54
CTNNB1 P35222 2/20 0.54
EGFR P00533 1/20 0.54
FGFR1 P11362 1/20 0.54
KDR P35968 1/20 0.54
BDKRB1 P46663 1/20 0.53
MAPT P10636 1/20 0.53
OPRM1 P35372 1/20 0.52
OPRD1 P41143 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17331311 0.91 KDM1A (0.70) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL17331331 0.90 LMNA (0.60) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL17331308 0.87 KMT2A (0.50) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL17347406 0.84 LMNA (0.74) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL17347484 0.84 ALDH1A1 (0.63) MEN1KMT2ALMNAHPGDMAPT
SCHEMBL17347396 0.82 ALDH1A1 (0.58) MEN1KMT2AHPGDBDKRB1MAPT
SCHEMBL8367822 0.82 KDM1A (0.60) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL8369354 0.80 TCF4 (0.80) MEN1KMT2ALMNAHDAC2HDAC8
SCHEMBL8699498 0.80 KDM1A (0.63) KDM1AMAOAMEN1KMT2ALMNA
SCHEMBL17331333 0.80 BDKRB1 (0.51) MEN1KMT2ABDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023076404-A1 METHODS FOR TREATING SYSTEMIC LUPUS ERYTHEMATOSUS ARIA PHARMACEUTICALS, INC. (US) 2023-05-04 WO disclosed
WO-2023076404-A1 METHODS FOR TREATING SYSTEMIC LUPUS ERYTHEMATOSUS ARIA PHARMACEUTICALS, INC. (US) 2023-05-04 WO disclosed
US-10004751-B2 Compositions and methods for treating Dengue virus infection THE J. DAVID GLADSTONE INSTITUTES (US) 2018-06-26 US disclosed
US-20170209460-A1 COMPOSITIONS AND METHODS FOR TREATING DENGUE VIRUS INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2017-07-27 US disclosed
US-9701627-B2 LRRK2 GTP binding inhibitors for treatment of Parkinson's disease and neuroinflammatory disorders UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-07-11 US disclosed
US-20150361038-A1 LRRK2 GTP BINDING INHIBITORS FOR TREATMENT OF PARKINSON'S DISEASE AND NEUROINFLAMMATORY DISORDERS UNIVERSITY OF MARYLAND, BALTIMORE 2015-12-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150361038-A1 LRRK2 GTP BINDING INHIBITORS FOR TREATMENT OF PARKINSON'S DISEASE AND NEUROINFLAMMATORY DISORDERS LRRK2, PARK7, SNCA KDM1A 4394/4885MAOA 3579/4885MEN1 4396/4885
US-10004751-B2 Compositions and methods for treating Dengue virus infection C5, HAVCR2, MAVS KDM1A 1987/4885MAOA 1411/4885MEN1 3171/4885
US-20170209460-A1 COMPOSITIONS AND METHODS FOR TREATING DENGUE VIRUS INFECTION C5, HAVCR2, MAVS KDM1A 1987/4885MAOA 1411/4885MEN1 3171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.