SCHEMBL17360435

SCHEMBL17360435

O=C1NC(=O)c2ccc3c4ccc5c6c(ccc(c7ccc1c2c73)c64)C(=O)NC5=O.O=S(=O)(O)c1ccccc1.O=S(=O)(O)c1ccccc1

nearest known ligand 0.52

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.52
TSHR P16473 1/20 0.52
GSK3B P49841 1/20 0.39
POLB P06746 3/20 0.39
PARP1 P09874 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CASP7 P55210 2/20 0.39
RGS12 O14924 1/20 0.39
USP2 O75604 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
CYP2C9 P11712 1/20 0.39
APEX1 P27695 1/20 0.39
CASP1 P29466 1/20 0.39
BRCA1 P38398 1/20 0.39
MTOR P42345 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalimide SCHEMBL30722317 0.83 SMN1; SMN2 (0.64) SMN1; SMN2TSHRGSK3BPOLBPARP1
Phthalimide SCHEMBL219747 0.83 SMN1; SMN2 (0.64) SMN1; SMN2TSHRGSK3BPOLBPARP1
SCHEMBL30606639 0.78 PARP1 (0.50) GSK3BPOLBPARP1MEN1KMT2A
SCHEMBL29541 0.78 PARP1 (0.50) GSK3BPOLBPARP1MEN1KMT2A
SCHEMBL7598089 0.78 PARP1 (0.50) GSK3BPOLBPARP1MEN1KMT2A
SCHEMBL7601076 0.78 PARP1 (0.50) GSK3BPOLBPARP1MEN1KMT2A
SCHEMBL5364036 0.78 CDK5 (0.45) TSHRPOLBPARP1MEN1KMT2A
SCHEMBL218236 0.76 SMN1; SMN2 (0.46) SMN1; SMN2TSHRGSK3BPOLBPARP1
SCHEMBL115116 0.72 TSHR (0.48) SMN1; SMN2TSHRGSK3BPOLBMEN1
SCHEMBL2509 0.72 TSHR (1.00) SMN1; SMN2TSHRPOLBTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960205-A1 Stable aqueous graphene suspension and its use in producing graphene polymer nanocomposites Solvay SA (BE) 2015-12-30 EP claimed
EP-2960205-A1 Stable aqueous graphene suspension and its use in producing graphene polymer nanocomposites Solvay SA (BE) 2015-12-30 EP disclosed