Capadenoson

Capadenoson

SCHEMBL174016

N#Cc1c(N)nc(SCc2csc(-c3ccc(Cl)cc3)n2)c(C#N)c1-c1ccc(OCCO)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1

The experimentally established mechanism targets of Capadenoson. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 known ✓ P30542 20/20 1.00
SLC6A3 Q01959 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3299665 0.92 ADORA1 (0.86) ADORA1SLC6A3
SCHEMBL13998935 0.92 ADORA1 (0.85) ADORA1SLC6A3
SCHEMBL1932981 0.92 ADORA1 (0.85) ADORA1SLC6A3
SCHEMBL20211460 0.92 ADORA1 (0.85) ADORA1SLC6A3
SCHEMBL14464879 0.91 ADORA1 (0.84) ADORA1SLC6A3
SCHEMBL7972583 0.91 ADORA1 (0.84) ADORA1SLC6A3
SCHEMBL1177603 0.91 ADORA1 (0.83) ADORA1SLC6A3
SCHEMBL7602052 0.91 ADORA1 (0.83) ADORA1SLC6A3
SCHEMBL3697062 0.90 ADORA1 (0.82) ADORA1SLC6A3
SCHEMBL14632034 0.90 ADORA1 (0.82) ADORA1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 198 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120114604-A Application of adenosine and receptor thereof in cardiopulmonary and cerebral resuscitation and multi-organ injury 中南大学湘雅医院 2025-06-10 CN claimed
EP-4178948-A2 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF Universidade de Santiago de Compostela (ES) 2023-05-17 EP claimed
WO-2017137528-A1 ADENOSINE A1 RECEPTOR AGONIST FOR USE IN TREATMENT OF STATUS EPILEPTICUS CHARITÉ - UNIVERSITÄTSMEDIZIN BERLIN (DE) 2017-08-17 WO claimed
US-20160311812-A1 ADENOSINE A1 AGONISTS AS MEDICAMENTS FOR KIDNEY DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-27 US claimed
WO-2013049725-A2 METHODS OF USING ADENOSINE A1 RECEPTOR ACTIVATION FOR TREATING DEPRESSION TUFTS UNIVERSITY (US) 2013-04-04 WO claimed
US-20080306070-A1 Combination Therapy Comprising Substituted Oxazolidinones for the Prevention and Treatment of Cerebral Circulatory Disorders BAYER HEALTHCARE AG 2008-12-11 US claimed
EP-1933841-A1 COMBINATION THERAPY COMPRISING SUBSTITUTED OXAZOLIDINONES FOR THE PREVENTION AND TREATMENT OF CEREBRAL CIRCULATORY DISORDERS Bayer HealthCare AG (DE) 2008-06-25 EP claimed
WO-2007039134-A1 COMBINATION THERAPY COMPRISING SUBSTITUTED OXAZOLIDINONES FOR THE PREVENTION AND TREATMENT OF CEREBRAL CIRCULATORY DISORDERS BAYER HEALTHCARE AG (DE) 2007-04-12 WO claimed
CN-116710439-B Substituted pyrazolopiperidine carboxylic acids BAYER AG (DE) 2026-05-26 CN disclosed
CN-116829545-B Substituted pyrazolylpiperidine carboxylic acids 拜耳公司 2026-05-15 CN disclosed
US-20260125401-A1 BORON-CONTAINING RHO KINASE INHIBITORS PERCIPIAD, INC. (US) 2026-05-07 US disclosed
EP-2841109-B1 PRODRUGS OF HYDROXYL-COMPRISING DRUGS ASCENDIS PHARMA AS (DK) 2026-04-15 EP disclosed
US-12595247-B2 Substituted pyrazolo piperidine carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 2026-04-07 US disclosed
US-20250361282-A1 ATRIAL NATRIURETIC PEPTIDE ENGRAFTED ANTIBODIES BAYER AKTIENGESELLSCHAFT (DE) 2025-11-27 US disclosed
WO-2007039134-A1 COMBINATION THERAPY COMPRISING SUBSTITUTED OXAZOLIDINONES FOR THE PREVENTION AND TREATMENT OF CEREBRAL CIRCULATORY DISORDERS BAYER HEALTHCARE AG (DE) 2007-04-12 WO disclosed
US-20060217373-A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same BAYER HEALTHCARE AG (DE) 2006-09-28 US disclosed
US-7109218-B2 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same BAYER HEALTHCARE AG (DE) 2006-09-19 US disclosed
US-20050227972-A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same BAYER HEALTHCARE AG (DE) 2005-10-13 US disclosed
EP-1455785-A1 SUBSTITUTED 2-THIO-3,5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THE USE OF THE SAME Bayer HealthCare AG (DE) 2004-09-15 EP disclosed
WO-2003053441-A1 SUBSTITUTED 2-THIO-3,5-DICYANO-4-PHENYL-6-AMINOPYRIDINES AND THE USE OF THE SAME BAYER HEALTHCARE AG (DE) 2003-07-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050227972-A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same TPMT, QDPR, TUBB6 ADORA1 998/4885SLC6A3 215/4885
US-20080306070-A1 Combination Therapy Comprising Substituted Oxazolidinones for the Prevention and Treatment of Cerebral Circulatory Disorders OTC, SDHA, SDHB ADORA1 1133/4885SLC6A3 1807/4885
US-20060217373-A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same TPMT, QDPR, TUBB6 ADORA1 998/4885SLC6A3 215/4885
US-12595247-B2 Substituted pyrazolo piperidine carboxylic acids SSB, PDK4, FPR1 ADORA1 1029/4885SLC6A3 1384/4885
US-20260125401-A1 BORON-CONTAINING RHO KINASE INHIBITORS NTRK2, GRK6, GRK1 ADORA1 2774/4885SLC6A3 312/4885
US-20160311812-A1 ADENOSINE A1 AGONISTS AS MEDICAMENTS FOR KIDNEY DISORDERS ADORA1, ADORA2A, ADORA2B ADORA1 1/4885SLC6A3 1206/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.