SCHEMBL17433959

SCHEMBL17433959

CCC1C(=O)N(CC2CC2)C(=O)c2cc([N+](=O)[O-])ccc21

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.48
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALOX5 P09917 1/20 0.39
RPS6KA2 Q15349 1/20 0.38
CASP1 P29466 1/20 0.38
CASP3 P42574 1/20 0.38
CASP4 P49662 1/20 0.38
CASP7 P55210 1/20 0.38
CASP9 P55211 1/20 0.38
CASP6 P55212 1/20 0.38
KDM1A O60341 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2658862 0.79 ACHE (0.70) ACHEALOX5RPS6KA2CA12CA1
SCHEMBL17434421 0.69 ACHE (0.47) ACHEALOX5KDM1ACA12CA1
SCHEMBL17434296 0.69 CYP3A4 (0.53) MEN1KMT2ACASP3CA1CA2
SCHEMBL6207633 0.67 ALOX5 (0.62) ACHEALOX5RPS6KA2CA12CA1
SCHEMBL14017942 0.67 PTPRC (0.53) ACHEMEN1KMT2AALOX5CASP1
SCHEMBL30070354 0.67 ALOX5 (0.62) ACHEALOX5RPS6KA2CA12CA1
SCHEMBL5113994 0.65 KMT2A (0.50) ACHEMEN1KMT2ACASP6KDM1A
SCHEMBL8090142 0.65 ACHE (0.62) ACHEMEN1KMT2AALOX5RPS6KA2
SCHEMBL18422262 0.64 ACHE (0.41) ACHECASP6KDM1A
SCHEMBL18422001 0.64 GRIN2B (0.47) ACHEMEN1KMT2ACASP6KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834520-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-12-05 US disclosed
US-20160229814-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-08-11 US disclosed
EP-2975031-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2016-01-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160229814-A1 HETEROCYCLIC COMPOUND RORB, RORC, RORA ACHE 2584/4885MEN1 2706/4885KMT2A 234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.