SCHEMBL17469335

SCHEMBL17469335

COc1ccc(-c2cc(C)c(C(C)=O)c(/C=C/c3ccccc3)c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.48
CYP1B1 Q16678 2/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1A2 P05177 1/20 0.46
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
MAOB P27338 2/20 0.45
HSPD1 P10809 1/20 0.45
TNFRSF1A P19438 1/20 0.45
HSPE1 P61604 1/20 0.45
CYP3A4 P08684 2/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TRPV1 Q8NER1 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17459512 0.91 TRPA1 (0.49) TRPA1CYP1B1CYP1A1CYP1A2MEN1
SCHEMBL17459513 0.91 TRPA1 (0.49) TRPA1CYP1B1CYP1A1CYP1A2MEN1
SCHEMBL17469313 0.88 TTR (0.42) TRPA1ALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL17469394 0.88 BCHE (0.46) CYP1B1CYP1A1CYP1A2MEN1ALDH1A1
SCHEMBL17469392 0.87 CYP1B1 (0.42) CYP1B1CYP1A2ALDH1A1MAPTCYP3A4
SCHEMBL17469388 0.86 POLB (0.46) TRPA1CYP1B1CYP1A1CYP1A2MEN1
SCHEMBL17469356 0.85 BCL2L1 (0.38) TRPA1MAPTKDM4ESMN1; SMN2LMNA
SCHEMBL17469314 0.84 RELA (0.42) CYP1B1RELA
SCHEMBL17469387 0.80 RAB9A (0.45) TRPA1CYP1A2MEN1ALDH1A1MAPT
SCHEMBL17459520 0.79 BCL2L1 (0.46) TRPA1ALDH1A1MAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016013976-A1 METHOD OF FORMING A MULTI-SUBSTITUTED BENZENE COMPOUND NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2016-01-28 WO disclosed