Serine

Serine

SCHEMBL1747404

N[C@@H](CO)C(=O)O.O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Serine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(D)-Serine SCHEMBL31186649 1.00
Serine SCHEMBL28890911 1.00
Serine SCHEMBL10623299 1.00
Serine SCHEMBL28890910 1.00
(D)-Serine SCHEMBL43094 0.97
Serine SCHEMBL1332181 0.97
Serine SCHEMBL2023739 0.97 SLC1A1 (0.59)
(D)-Serine SCHEMBL6660617 0.97 SLC1A1 (0.59)
Serine SCHEMBL6929773 0.97 SLC1A1 (0.59)
Serine SCHEMBL2023740 0.97 SLC1A1 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343808-A2 PROCESS FOR THE SYNTHESIS OF A PEPTIDE HAVING A TRP RESIDUE Kinerton Limited (IE) 2003-09-17 EP claimed
WO-2002051861-A2 PROCESS FOR THE SYNTHESIS OF A PEPTIDE HAVING A TRYPTOPHAN RESIDUE KINERTON LIMITED (IE) 2002-07-04 WO claimed
JP-57035549-A None JP disclosed
JP-57032256-A None JP disclosed
JP-57035548-A None JP disclosed
CN-119707944-A Hydrated compound and preparation method thereof 福建省闽东力捷迅药业股份有限公司 2025-03-28 CN disclosed
EP-3293522-A2 LIPIDOMIC BIOMARKERS FOR IDENTIFICATION OF HIGH-RISK CORONARY ARTERY DISEASE PATIENTS Zora Biosciences OY (FI) 2018-03-14 EP disclosed
EP-2385374-B2 Lipidomic biomarkers for atherosclerosis and cardiovascular disease ZORA BIOSCIENCES OY (FI) 2018-02-28 EP disclosed
US-20160025751-A1 Lipidomic Biomarkers for Identification of High-Risk Coronary Artery Disease Patients ZORA BIOSCIENCES OY (FI) 2016-01-28 US disclosed
WO-2013012846-A1 PROCESS FOR PREPARING PHOSPHORYLATED AMINO ACIDS CEPHALON, INC. (US) 2013-01-24 WO disclosed
WO-2013012416-A1 PROCESS FOR PREPARING PHOSPHORYLATED AMINO ACIDS CEPHALON, INC. (US) 2013-01-24 WO disclosed
EP-2385374-A1 Lipidomic biomarkers for atherosclerosis and cardiovascular disease Zora Biosciences OY (FI) 2011-11-09 EP disclosed
US-8040688-B2 Circuit board unit and electronic device FUJITSU LIMITED (JP) 2011-10-18 US disclosed
US-4725645-A USING A TRIALKYLCYANOSILANE SOLVAY & CIE. (SOCIETE ANONYME) (BE) 1988-02-16 US disclosed
EP-0164389-B1 PREPARATION OF PHENYL ALANINES BY HYDROGENATION OF PHENYL SERINES ALKALOIDA VEGYéSZETI GYáR (HU) 1987-04-01 EP disclosed
EP-0164389-A1 PREPARATION OF PHENYL ALANINES BY HYDROGENATION OF PHENYL SERINES. ALKALOIDA VEGYESZETI GYAR (HU) 1985-12-18 EP disclosed
WO-1985002609-A1 PREPARATION OF PHENYL ALANINES BY HYDROGENATION OF PHENYL SERINES ALKALOIDA VEGYÉSZETI GYÁR (HU) 1985-06-20 WO disclosed
JP-S5735549-A OBTAINING METHOD OF AMINO ACID HYDRATE CRYSTAL AJINOMOTO CO INC 1982-02-26 JP disclosed
JP-S5735548-A DRYING METHOD OF AMINO ACID CRYSTAL AJINOMOTO CO INC 1982-02-26 JP disclosed
JP-S5732256-A CRYSTALLIZATION OF SERINE AJINOMOTO CO INC 1982-02-20 JP disclosed