SCHEMBL1748172

SCHEMBL1748172

C[C@@]1(C(=O)O)CCC[C@H]1C(=O)c1ccc(-c2ccc(N)c(F)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.36
HDAC1 Q13547 6/20 0.36
HDAC3 O15379 5/20 0.36
HDAC2 Q92769 5/20 0.36
HDAC6 Q9UBN7 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CTSL P07711 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
PDE4D Q08499 1/20 0.34
RARA P10276 2/20 0.33
RARB P10826 2/20 0.33
RARG P13631 2/20 0.33
KIF11 P52732 1/20 0.33
HSD11B1 P28845 1/20 0.32
APP P05067 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2311893 0.85 NPC1 (0.35) DGAT1HSD17B10PDE4DRARARARB
SCHEMBL2309580 0.83 DGAT1 (0.41) DGAT1KDM4ELMNAHSD17B10PDE4D
SCHEMBL1748043 0.79 ALDH1A1 (0.38) HDAC1HDAC3HDAC2KDM4ELMNA
SCHEMBL1748045 0.79 ALDH1A1 (0.38) HDAC1HDAC3HDAC2KDM4ELMNA
SCHEMBL1748044 0.79 ALDH1A1 (0.38) HDAC1HDAC3HDAC2KDM4ELMNA
SCHEMBL2635426 0.74 DGAT1 (0.60) DGAT1HDAC1HDAC6
SCHEMBL4923255 0.74 HSD17B1 (0.39) HDAC1HDAC3HDAC2KDM4E
SCHEMBL1748065 0.74 DGAT1 (0.41) DGAT1HDAC6KDM4EHSD17B10
SCHEMBL14074139 0.73 DGAT1 (0.46) DGAT1HDAC1HDAC3HDAC2HDAC6
SCHEMBL1748238 0.73 DGAT1 (0.42) DGAT1HDAC6KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8013166-B2 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER HEALTHCARE LLC (US) 2011-09-06 US disclosed
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP disclosed